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    當前位置:首頁 > 技術文章 > levenabiopharma產品目錄

    levenabiopharma產品目錄

    更新時間:2021-01-08      點擊次數:1659

     

     levenabiopharma用于連接抗體和藥物的連接子

    levenabiopharma生物制藥提供不同結構和功能的多種連接子,可用于抗體和藥物的偶聯的連接子。更重要的是,聯寧自主開發的擁有*知識產權的連接子可以將藥物可控地偶聯到抗體上,更易實現批次間的產品質量控制。為更好地支持客戶的藥物開發,levenabiopharma還提供連接子定制設計和合成服務。

    levenabiopharma產品目錄

     

    產品目錄號產品名稱Cas 號純度可提供數量
    VC1001Val-Cit-PAB159857-79-195%mg - 500g
    VC1002Fmoc-Val-Cit-PAB159858-22-795%mg - 500g
    VC1003Fmoc-Val-Cit-PAB-PNP863971-53-395%mg - 500g
    VC1004MC-Val-Cit-PAB-PNP159857-81-595%mg-100g
    FK1001Phe-Lys(Trt)-PAB 95%mg - kg
    FK1002Fmoc-Phe-Lys(Trt)-PAB 95%mg - kg
    FK1003Fmoc-Phe
    -Lys(Trt)-PAB-PNP
    1116086-09-995%mg - kg
    AN1001Ala-Ala-Asn-PAB TFA salt 95%mg - kg
    AN1002Fmoc-Ala-Ala-Asn-PAB-PNP 95%mg - kg
    H1001Fmoc-Gly3-Val-Cit-PAB 95%mg-100g
    H1002Fmoc-Gly3-Val-Cit-PAB-PNP 95%mg-100g
    D1000SMCC64987-85-598%500mg-500g
    DS1001Py-ds-Prp-OSu 95%mg - kg
    DS1003Py-ds-dmBut-OSu 95%mg - 100g
    DS1013Py-ds-dmBut-OPFP 95%mg - 100g
    DS1011Py-ds-Prp-OPFP 95%mg - kg
    MA1000MAL-HA-OSu 95%mg - kg
    MA2011MAL-di-EG-OPFP 95%mg - kg
    MA2012MAL-tri-EG-OPFP 95%mg - kg
    MA2013MAL-tetra-EG-OPFP 95%mg - kg
    AZ1011N3-di-EG-OPFP 95%mg - kg
    AZ1012N3-tri-EG-OPFP 95%mg - kg
    AZ1013N3-tetra-EG-OPFP 95%mg - kg
    AL1001ALD-BZ-OSu 95%mg - kg
    AL1003ALD-di-EG-OSu 95%mg - kg
    AL1005ALD-tetra-EG-OSu 95%mg - kg
    AL1013ALD-di-EG-OPFP 95%mg - kg
    AL1015ALD-tetra-EG-OPFP 95%mg - kg
    HA1011PHA-di-EG-OPFP 95%mg - kg
    HA1013PHA-tetra-EG-OPFP 95%mg - kg

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    ADC細胞毒素藥物

     

    從抗體到靶向抗體藥物偶聯物的合成過程有挑戰性。為了設計出高效的抗體藥物偶聯物,毒素的選擇是至關重要的。聯寧生物制藥提供各種各樣的微管蛋白抑制劑和DNA烷基化試劑,這些試劑已被證實是抗體藥物偶聯物負載的有效細胞毒素。對下面列出的這些毒素, 聯寧可以提供毫克級至100克級的高質量產品。

    For structures, click here>>>

    產品目錄號產品名稱Cas 號純度可提供數量
    T1001Dolastatin 10110417-88-498%mg - 100g
    T1002Monomethyl Dolastatin 10203849-91-698%mg - 100g
    T1003Auristatin E160800-57-798%mg - 100g
    T1004Monomethyl Auristatin E474645-27-798%mg - 100g
    T1005Auristatin F163768-50-198%mg - 100g
    T1006Monomethyl Auristatin F745017-94-198%mg - 100g
    T1007HTI-286228266-40-895%mg - g
    T1008Tubulysin M205304-86-595%mg - g
    T1009Maytansinoid AP-366547-09-985%mg
    T1109Maytansinol57103-68-195%mg - 100g
    LN-T-4582DM1139504-50-098%mg - 100g
    LN-T-7544DM4799840-96-398%mg - 10g
    T1102Boc-Val-Dil-Dap-OH 95%mg - kg
    T1202Boc-Val-Dil-Dap-Phe-OMe 95%mg - kg
    T1222Boc-Val-Dil-Dap-Doe 95%mg - kg
    T1224Boc-Val-Dil-Dap-Nrp 95%mg - kg
    T1302Boc-N-Me-Val-Val-Dil-Dap-OH 95%mg - kg
    T1108Tubulysin IM-1 95%mg - 100g
    T1208Tubulysin IM-2 95%mg - 100g
    T1308Tubulysin IM-3 95%mg - 100g
    D1001Duocarmycin SA152785-82-595%mg - g
    D1007Duocarmycin TM 95%mg - g
    D1008Duocarmycin MA 95%mg - g
    D1009Duocarmycin DM 95%mg - g
    D4000Nemorubicin108852-90-095%mg - 10 g
    D4001PNU-159682202350-68-3>90%mg -10 g
    LN-T-6888Calicheamicin g1108212-75-5>95%mg-100mg
    D4006N-Acetyl-Calicheamicin g1108212-76-6
    >95%
    mg-100g
    D4007a-Amanitin23109-05-9>95%mg-g
    D4008PBD-dimer1222490-34-7>90%mg-100mg

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    易用的細胞毒素 (SET™)

    聯寧生物制藥提供安全易用的毒素(SET™),這是一種可以快速篩選抗體藥物偶聯物的新型研究工具。SET™產品線包括很多已驗證的連接子-毒素,分別裝入預包裝好的小瓶中。每個SET™小瓶含有約200納摩的連接子-毒素,按藥物/抗體比(DAR)為3-4計算的話, 足夠偶聯5毫克抗體。客戶不需要稱重或分裝連接子-毒素,只需按照產品說明書上提供的溶解方案,即可使用SET™。SET™不僅易于使用,更重要的是可以大限度地減少實驗過程中暴露毒素的風險。目前,SET™可用于以下類別的偶聯反應:

     

        ?胺反應SET™ 
        ?硫醇反應SET™ 
        ?點擊反應SET™ 
        ?轉肽酶反應 SET™ 

    For structures, click here>>>

    胺反應 SET™  
    產品目錄號產品名稱數量單價
    SET0100OSu-Glu-vc-PAB-MMAE200 nmol$500
    SET0101SMCC-DM1200 nmol$500
    SET0102SPDB-DM4200 nmol$650
    SET0103OSu-PEG4-vc-PAB-DMEA
    Duocarmycin SA
    200 nmol$750
    SET0104Mylotarg-linker200 nmol$950
    SET0105OSu-Glu-vc-PAB-MMAD200 nmol$500
    SET0106Sulfo-SPDB-DM4200 nmol$950.00
    SET0107IMGN779-linker200 nmol$2,200.00
    SET0108OSu-PEG4-vc-PAB-DMEA
    Duocarmycin TM
    200 nmol$750.00
    SET0109OSu-PEG4-vc-PAB-DMEA
    Duocarmycin DM
    200 nmol$750.00
    硫醇反應SET™  
    產品目錄號產品名稱數量單價
    SET0201MC-vc-PAB-MMAE200 nmol$ 500
    SET0202MC-MMAF200 nmol$ 500
    SET0203MC-DM1200 nmol$ 700
    SET0204MC-MMD-10200 nmol$ 600
    SET0205MA-PEG4-vc-PAB-DMEA-
    duocarmycin SA
    200 nmol$ 750
    SET0206MC-vc-PAB-C6-a-amanitin200 nmol$ 850
    SET0207MC-cleavable-linker-a-amanitin200 nmol$ 600
    SET0208MC-vc-PAB-DMEA-(PEG2)-
    duocarmycin SA
    200 nmol$ 800
    SET0209MC-vc-PAB-Tubulysin M200 nmol$ 800
    SET0210MC-va-PAB-MMAD200 nmol$ 500
    SET0211MA-PEG4-VC-PAB-DMAE-PNU159682200 nmol$ 950
    SET0212MA-PEG4-VA-PBD200 nmol$ 1,100
    SET0213MC-vc-PAB-MMAF200 nmol$ 500
    SET0214MC-vc-PAB-MMAD200 nmol$ 500
    SET0215MC-vc-PAB-Auristatin 0101200 nmol$ 900
    SET0216MA-PEG8-VA-PAB-SG3199200 nmol$ 1,950
    SET0217CL2A-SN 38200 nmol$ 800
    SET0218MC-GGFG-DX8951200 nmol$ 950
    SET0219MEDI4276_linker payload200 nmol$ 1,100
    SET0220MA-PEG4-vc-PAB-DMEA-
    duocarmycin TM
    200 nmol$ 750
    SET0221MC-vc-PAB-(PEG2)-
    duocarmycin TM
    200 nmol$ 900
    SET0222MA-PEG4-vc-PAB-DMEA-
    duocarmycin DM
    200 nmol$ 750
    SET0223MC-vc-PAB-(PEG2)-
    duocarmycin DM
    200 nmol$ 900
    SET0224DGN549200 nmol$ 1,900
    SET0225MPB-vc-PAB-MMAE200 nmol$ 550
    SET0226MPB-MMAF200 nmol$ 550
    點擊反應SET™  
    產品目錄號產品名稱數量單價
    SET0301DBCO-PEG4-vc-PAB-MMAE200 nmol$ 650
    SET0302DBCO-PEG4-MMAF200 nmol$ 750
    SET0303DBCO-PEG4-Ahx-DM1200 nmol$ 750
    SET0304DBCO-PEG4-vc-PAB-
    Duocarmycin SA
    200 nmol$ 900
    SET0305DBCO-PEG4-vc-PAB-(PEG2)-
    Duocarmycin SA
    200 nmol$ 1,050
    SET0306DBCO-PEG4-VA-PBD200 nmol$ 1,100
    SET0307DBCO-PEG4-vc-PAB-MMAF200 nmol$ 650
    SET0308DBCO-PEG4-vc-PAB-MMAD200 nmol$ 650
    SET0309DBCO-PEG4-vc-PAB-
    Duocarmycin TM
    200 nmol$ 900
    SET0310DBCO-PEG4-vc-PAB-(PEG2)-
    Duocarmycin TM
    200 nmol$ 1,050
    SET0311DBCO-PEG4-vc-PAB-
    Duocarmycin DM
    200 nmol$ 900
    SET0312DBCO-PEG4-vc-PAB-(PEG2)-
    Duocarmycin DM
    200 nmol$ 1,050
    SET0313DBCO-PEG4-VC-PAB-DMAE-PNU159682200 nmol$ 1,050
    SET0314DBCO-PEG4-DMAE-PNU159682200 nmol$ 1,000
    SET0315DBCO-PEG4-GGFG-DX8951200 nmol$ 1,050
    SET0316DBCO-PEG4-vc-PAB-Ahx-DM1200 nmol$ 850
    SET0317DBCO-PEG8-VA-PAB-SG3199200 nmol$ 2,050
    轉肽酶反應 SET™  
    產品目錄號產品名稱數量單價
    SET0401Gly3-vc-PAB-MMAE200 nmol$850
    SET0402Gly3-MMAF200 nmol$850
    SET0403Gly5-Ahx-DM1200 nmol$950
    SET0404PNU159682-EDA-Gly3200 nmol$1,100

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    ADC篩選試劑盒

     

     

    聯寧生物制藥提供研究階段抗體藥物偶聯物體外活性的篩選服務。公司的細胞庫擁有超過100個癌細胞株,可以幫助客戶評估抗體藥物偶聯物的細胞毒性和治療潛力。公司還可以根據客戶的需求靈活安排用這些細胞株來篩選抗體藥物偶聯物。

     

    聯寧生物制藥制備了目前市面上常用的抗體藥物偶聯物,如T-DM1,brentuximab vedotin,VEGR2-ADC等,作為抗體藥物偶聯物評估的對照物,為客戶評估抗體藥物偶聯物生物仿制藥提供方便。

    聯寧生物制藥開發的以蛋白A和蛋白G的PSKA™和PSKG™的抗體藥物偶聯物預篩選試劑盒,在不做偶聯的情況下, 可以快速鑒定適合抗體藥物偶聯物研發用的抗體。使用這些試劑盒,可以直接篩選初級抗體,略去單獨將毒素偶聯到抗體上的過程。我們提供的PSK篩選試劑盒包括業界常用毒素,如MMAE,MMAF,DM1和duocarmycin。

    產品目錄號產品名稱產品說明數量單價
    LEV-PSKA-100ADC pre-screening kit AFour vials containing Protein A preloaded with
    1x MMAE (cleavable linker) 
    1x MMAF (non-cleavable linker) 
    1x MCC-DM1 (non-cleavable linker)
    1x Duocarmycin (cleavable linker)
    4x100 µL$ 900.00
    LEV-ADM-100Protein A-DM1Protein A preloaded with MCC-DM1 (non-cleavable linker)100 µL$ 300.00
    LEV-AME-100Protein A-MMAEProtein A preloaded with MMAE (cleavable linker)100 µL$ 300.00
    LEV-AMF-100Protein A-MMAFProtein A preloaded with MMAF (non-cleavable linker)100 µL$ 300.00
    LEV-ADC-100Protein A-DuocarmycinProtein A preloaded with Duocarmycin (cleavable linker)100 µL$ 400.00
    LEV-ACC-100Protein A-CalicheamicinProtein A preloaded with Calicheamicin (cleavable linker)100 µL$ 400.00
    LEV-APB-100Protein A-PBDProtein A preloaded with PBD100 µL$ 400.00
    LEV-PSKG-100ADC pre-screening kit GFour vials containing Protein A preloaded with
    1x MMAE (cleavable linker) 
    1x MMAF (non-cleavable linker) 
    1x MCC-DM1 (non-cleavable linker)
    1x Duocarmycin (cleavable linker)
    4x100 µL$ 900.00
    LEV-GDM-100Protein G-DM1Protein G preloaded with MCC-DM1 (non-cleavable linker)100 µL$ 300.00
    LEV-GME-100Protein G-MMAEProtein G preloaded with MMAE (cleavable linker)100 µL$ 300.00
    LEV-GMF-100Protein G-MMAFProtein G preloaded with MMAF (non-cleavable linker)100 µL$ 300.00
    LEV-GDC-100Protein G-DuocarmycinProtein G preloaded with Duocarmycin (cleavable linker)100 µL$ 400.00
    LEV-GAM-100Protein G-AmanitinProtein G preloaded with Amanitin (cleavable linker)100 µL$ 400.00
    LEV-GAL-100Protein G-AmanitinProtein G preloaded with Amanitin (Levena cleaveable linker)100 µL$ 400.00

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    抗細胞毒性藥物抗體

     

     

    聯寧生物制藥開發了各種抗細胞毒性藥物抗體用來支持客戶的臨床前藥物研究。目前,提供的抗體包括針對不同類別的細胞毒性藥物的抗毒素(藥物)單克隆和多克隆抗體。這些產品僅限于科研,不能用于臨床診斷

    產品目錄號產品名稱毒素類型微升單價毫克/毫升
    LEV-PAE1-100Rabbit Anti-vc-PAB-MMAE pAbTubulin Inhibitor100 $    500.001
    LEV-PAE1-500500 $ 1,875.00
    LEV-MAE1-100Mouse Anti-vc-PAB-MMAE mAb (B11F11)Tubulin Inhibitor100 $    900.001
    LEV-MAE1-500500 $ 3,375.00
    LEV-PAF1-100Rabbit Anti-MMAF pAbTubulin Inhibitor100 $    500.001
    LEV-PAF1-500500 $ 1,875.00
    LEV-MAF1-100Mouse Anti-MMAF mAb (F3B11)Tubulin Inhibitor100 $    900.001
    LEV-MAF1-500500 $ 3,375.00
    LEV-MAE3-100Mouse Anti-MMAE / F mAb (B12A2)Tubulin Inhibitor100 $    900.001
    LEV-MAE3-500500 $ 3,375.00
    LEV-MAF3-100Mouse Anti-MMAE /F mAb (C12A1)Tubulin Inhibitor100 $    900.001
    LEV-MAF3-500500 $ 3,375.00
    LEV-PDM1-100Rabbit Anti-DM1/4 pAbTubulin Inhibitor100 $    500.001
    LEV-PDM1-500500 $ 1,875.00
    LEV-MDM1-100Mouse Anti-DM1/4 mAb (F1D5)Tubulin Inhibitor100 $    900.001
    LEV-MDM1-500500 $ 3,375.00
    LEV-MDM2-100Mouse Anti-DM1/4 mAb (G2F3)Tubulin Inhibitor100 $    900.001
    LEV-MDM2-500500 $ 3,375.00
    LEV-PCA1-100Rabbit Anti-Calicheamicin pAbDNA Damaging100 $    750.000.5
    LEV-PCA1-500500 $ 2,800.00
    LEV-MCA1-100Mouse Anti-Calicheamicin mAb (B1G9)DNA Damaging100 $ 1,250.000.5
    LEV-MCA1-500500 $ 4,700.00
    LEV-MCA2-100Mouse Anti-Calicheamicin mAb (C1F12) DNA Damaging100 $ 1,250.000.5
    LEV-MCA2-500500 $ 4,700.00
    LEV-PDU1-100Rabbit Anti-Duocarmycin pAb DNA Damaging100 $    750.000.5
    LEV-PDU1-500500 $ 2,800.00
    LEV-MDU3-100Mouse Anti-Duocarmycin mAb (E11A1) DNA Damaging100 $    900.000.5
    LEV-MDU3-500500 $ 3,375.00
    LEV-MDU1-100Mouse Anti-Duocarmycin mAb (H7A9)DNA Damaging100 $    900.000.5
    LEV-MDU1-500500 $ 3,375.00
    LEV-MDU2-100Mouse Anti-Duocarmycin mAb (E6B3) DNA Damaging100 $    900.000.5
    LEV-MDU2-500500 $ 3,375.00
    LEV-PPN1-100Rabbit Anti-PNU-159682 pAbDNA Damaging100 $    750.000.5
    LEV-PPN1-500500 $ 2,800.00
    LEV-MPN1-100Mouse Anti-PNU-159682 mAb (F7F2)DNA Damaging100 $    900.000.5
    LEV-MPN1-500500 $ 3,375.00
    LEV-MPN2-100Mouse Anti-PNU-159682 mAb (C1E3)DNA Damaging100 $    900.000.5
    LEV-MPN2-500500 $ 3,375.00
    LEV-MPN3-100Mouse Anti-PNU-159682 mAb (D12H11)DNA Damaging100 $    900.000.5
    LEV-MPN3-500500 $ 3,375.00
    LEV-PAM1-100Rabbit Anti-Amanitin pAbRNA Polymerase II and III Inhibitor100 $    650.000.5
    LEV-PAM1-500500 $ 2,450.00
    LEV-MAM1-100Mouse Anti-Amanitin mAb (H3E1)RNA Polymerase II and III Inhibitor100 $ 1,100.000.5
    LEV-MAM1-500500 $ 4,100.00
    LEV-MAM2-100Mouse Anti-Amanitin mAb (H12D6)RNA Polymerase II and III Inhibitor100 $ 1,100.000.5
    LEV-MAM2-500500 $ 4,100.00
    LEV-MAM3-100Mouse Anti-Amanitin mAb (C2C4)RNA Polymerase II and III Inhibitor100 $ 1,100.000.5
    LEV-MAM3-500500 $ 4,100.00
    LEV-PSN1-100Rabbit Anti-SN38 pAbDNA Topoisomerase I Inhibitor100 $    650.000.5
    LEV-PSN1-500500 $ 2,450.00
    LEV-MSN1-100Mouse Anti-SN38 mAb (10F11A9D6)DNA Topoisomerase I Inhibitor100 $    900.000.5
    LEV-MSN1-500500 $ 3,375.00
    LEV-MSN2-100Mouse Anti-SN38 mAb (8E10F12F3)DNA Topoisomerase I Inhibitor100 $    900.000.5
    LEV-MSN2-500500 $ 3,375.00
    LEV-MSN3-100Mouse Anti-SN38 mAb (8E10A4A1)DNA Topoisomerase I Inhibitor100 $    900.000.5
    LEV-MSN3-500500 $ 3,375.00
    LEV-PSG1-100Rabbit Anti-PBD SG3199 pAb DNA Inhibitor                                100 $    900.000.5
    LEV-PSG1-500500 $ 3,374.00
    LEV-MSG1-100Mouse Anti-PBD SG3199 (7H6H9A6) mAbDNA Inhibitor100 $ 1,250.000.5
    LEV-MSG1-500500 $ 4,500.00
    LEV-MSG2-100Mouse Anti-PBD SG3199 (8G2H12A9) mAbDNA Inhibitor100 $ 1,250.000.5
    LEV-MSG2-500500 $ 4,500.00
    LEV-MSG3-100Mouse Anti-PBD SG3199 (8B3D12G1) mAbDNA Inhibitor100 $ 1,250.000.5
    LEV-MSG3-500500 $ 4,500.00

     

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